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GLP-1 comparison

Retatrutide vs tirzepatide

Retatrutide is the newer triple-agonist; tirzepatide is the established dual-agonist. They differ in mechanism and in how far along they are, which is worth understanding before you compare doses. This page lays out the facts and links each calculator.

DimensionRetatrutideTirzepatide
ClassGLP-1 / GIP / glucagon agonistGLP-1 / GIP agonist
CategoryGLP-1GLP-1
Common vial sizes5 / 10 mg5 / 10 / 15 mg
Typical dose range1 mg – 12 mg2.5 mg – 15 mg
Half-life~6 days~5 days
StatusResearch compoundFDA-approved formulation exists

Educational reference only. Not medical advice — follow the instructions from your clinician or pharmacy.

Triple vs dual agonist

Retatrutide targets three receptors (GLP-1, GIP, and glucagon); tirzepatide targets two (GLP-1 and GIP). The extra glucagon activity is the headline difference and is why retatrutide is studied at its own dose range rather than tirzepatide's.

For reconstitution, both are handled the same way — only the milligram numbers and vial sizes differ, as the table above shows.

  • Retatrutide: GLP-1 + GIP + glucagon (triple)
  • Tirzepatide: GLP-1 + GIP (dual)
  • Separate dose ranges — not interchangeable

Maturity and how it affects sourcing

Tirzepatide has an approved formulation; retatrutide is still investigational. That difference does not change the calculator math, but it does mean retatrutide doses come from research vials rather than an approved product, so confirm your vial strength carefully before calculating.

Whichever you use, run your real vial and water numbers through the relevant calculator to get the exact draw.

Frequently asked questions

Is retatrutide stronger than tirzepatide?+
They are different molecules with different receptor targets and separate dose ranges, so 'stronger' is not a simple comparison. This page compares their facts for context only and does not recommend doses.
Can I convert a tirzepatide dose to retatrutide?+
No — the dose ranges are studied independently and do not convert one-to-one. Use the dose your protocol specifies for the specific compound, then calculate the draw on that compound's page.
Is the reconstitution the same for both?+
Yes, the math is identical; only the vial sizes and milligram doses differ. The table above shows those differences, pulled from the same data the calculators use.
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